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(+)-CGP-12177A

(+)-CGP-12177A is a synthetic hydrophilic inhibitor of the adrenergic receptors β1, β2, and β3 (Ki=0.9, 4, and 88nM, respectively). Inhibits isoproterenol stimulation of adenylyl cyclase activity at low concentrations. Can also act as an agonist of these receptors at higher concentrations.

Catalog No. Size Price Quantity
92-1216 10 mg $108.00

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Description
(+)-CGP-12177A
Compound Type
Agonist
Storage
RT
Source
Synthetic
Cells were plated in a 384-well plate and incubated overnight at 37°C/5% CO2 to allow the cells to attach and grow. Cells were then stimulated with a control agonist, using the assay conditions described below. Following stimulation, signal was detected using the HitHunter cAMP Assay Detection Kit according to the recommended protocol.