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Alphabetical Target List

AAK1 ABL1 ABL1(E255K)-phosphorylated ABL1(F317I)-nonphosphorylated ABL1(F317I)-phosphorylated
ABL1(F317L)-nonphosphorylated ABL1(F317L)-phosphorylated ABL1(H396P)-nonphosphorylated ABL1(H396P)-phosphorylated ABL1(M351T)-phosphorylated
ABL1(Q252H)-nonphosphorylated ABL1(Q252H)-phosphorylated ABL1(T315I)-nonphosphorylated ABL1(T315I)-phosphorylated ABL1(Y253F)-phosphorylated
ABL1-nonphosphorylated ABL1-phosphorylated ABL2 ACVR1 ACVR1B
ACVR1B/BMPR2 ACVR1C/ACVR2 ACVR1C/ACVR2B ACVR2/ACVR1 ACVR2A
ACVR2B ACVRL1 ACVRL1/ACVR2 ACVRL1/ACVR2B ACVRL1/BMPR2
ADCK3 ADCK4 ADCYAP1R1 ADORA1 ADORA2A
ADORA2B ADORA3 ADRA1A ADRA1B ADRA1D(82-572)
ADRA2A ADRA2B ADRA2C ADRB1 ADRB2
ADRB2(W158A) ADRB3 AGTR1 AGTRL1 AKT1
AKT2 AKT3 ALK ALK(1151Tins) ALK(C1156Y)
ALK(F1174L) ALK(L1196M) AMPK-alpha1 AMPK-alpha2 ANKK1
AR ARK5 ASK1 ASK2 ATAD2A
ATAD2B ATAD2B AURKA AURKB AURKC
AVPR1A AVPR1B AVPR2 AVPR2(S167T) AXL
BAI1 BAI2 BAI3 BAZ2A BAZ2A
BAZ2B BCL2-BAX BCL2-BIM BCL2L1-BAX BCL2L1-BIM
BDKRB1 BDKRB2 BIKE BLK BMPR1A
BMPR1A/ACVR2 BMPR1A/ACVR2B BMPR1A/BMPR2 BMPR1B BMPR1B/ACVR2
BMPR1B/ACVR2B BMPR1B/BMPR2 BMPR2 BMX BRAF
BRAF(V600E) BRD1 Brd2(1) BRD2(1,2) BRD2(2)
BRD3(1) BRD3(1) BRD3(1,2) BRD3(2) Brd4(1)
BRD4(1,2) BRD4(2) BRD4(full-length,short-iso.) Brd7 BRD8(1)
BRD8(2) BRD9 BrdT(1) BRDT(1,2) BRDT(2)
BRK BRPF1 BRPF3 BRPF3 BRS3
BRSK1 BRSK2 BRWD3(2) BTK BUB1
C3AR1 C5AR1 C5L2 CALCR CALCRL-RAMP1
CALCRL-RAMP2 CALCRL-RAMP3 CALCR-RAMP2 CALCR-RAMP3 CAMK1
CAMK1B CAMK1D CAMK1G CAMK2A CAMK2B
CAMK2D CAMK2G CAMK4 CAMKK1 CAMKK2
CASK CASR CCKAR CCKBR CCR1
CCR10 CCR2 CCR3 CCR4 CCR5
CCR6 CCR7 CCR8 CCR9 CCRL1
CCRL2 CD137 CD86 CDC25A CDC2L1
CDC2L2 CDC2L5 CDK1 CDK10 CDK11
CDK12 CDK2 CDK20 CDK3 CDK4
CDK4-cyclinD1 CDK4-cyclinD1(F93L) CDK4-cyclinD3 CDK5 CDK6
CDK7 CDK8 CDK9 CDKL1 CDKL2
CDKL3 CDKL5 CECR2 cEDG5 CFTR-ΔF508
cGPR91 CHEK1 CHEK2 CHRM1 CHRM2
CHRM3 CHRM4 CHRM5 cINSRa cINSRb
CIT c-KIT CLK1 CLK2 CLK3
CLK4 c-MET/c-MET CMKLR1 CNR1 CNR2
CREBBP c-Ret-GFRα1 c-Ret-GFRα2 CRHR1 CRHR2
CRTH2 CSF1R CSF1R/CSF1R CSF1R-autoinhibited CSF2RB/CSF2RA
CSF3R-JAK1 CSK CSNK1A1 CSNK1A1L CSNK1D
CSNK1E CSNK1G1 CSNK1G2 CSNK1G3 CSNK2A1
CSNK2A2 CTK CTLA4 CX3CR1 CXCR1
CXCR2 CXCR3 CXCR4 CXCR5 CXCR6
CXCR7 cyno CXCR1 cyno CXCR2 cyno GPR120 cyno MRGPRX2
CYSLTR2 DAPK1 DAPK2 DAPK3 DARC
DCAMKL1 DCAMKL2 DCAMKL3 DDR1 DDR2(T654M)
DLK DMPK DMPK2 DRAK1 DRAK2
DRD1 DRD2L DRD2S DRD3 DRD4
DRD5 DYRK1A DYRK1B DYRK2 EBI2
EDG1 EDG2 EDG3 EDG4 EDG5
EDG6 EDG7 EDNRA EDNRB EGFR
EGFR(E746-A750del) EGFR(G719C) EGFR(G719S) EGFR(L747-E749del, A750P) EGFR(L747-S752del, P753S)
EGFR(L747-T751del,Sins) EGFR(L858R) EGFR(L858R,T790M) EGFR(L861Q) EGFR(S752-I759del)
EGFR(T790M) EGFR/EGFR EGFR/ErbB2 EGFR/ErbB3 EIF2AK1
EP300 EP300 EPHA1 EPHA2 EPHA3
EphA4 EphA5 EPHA6 EphA7 EPHA8
EphB1 EphB2 EphB3 EphB4 EPHB6
EpoR/EpoR EpoR-JAK2 ErbB1 ERBB2 ErbB2/ErbB3
ErbB2/ErbB4 ErbB2-ErbB3 ERBB3 ErbB4 ErbB4/ErbB4
ERK1 ERK1(Q122L) ERK2 ERK3 ERK4
ERK5 ERK8 ERN1 ERRα ERα
F2R F2RL1 F2RL3 FAK FALZ
FALZ FER FES FFAR1 FFAR2
FFAR3 FGFR1 FGFR1-α-Klotho FGFR1-β-Klotho FGFR2
FGFR2(N550K) FGFR3 FGFR3(G380R)/FGFR3(G380R) FGFR3(G697C) FGFR3(K650E)
FGFR3(V555M) FGFR3/FGFR3 FGFR4 FGFR4 FGFR4-α-Klotho
FGFR4-β-Klotho FGR FLT1 FLT3 FLT3(D835H)
FLT3(D835V) FLT3(D835Y) FLT3(ITD) FLT3(ITD,D835V) FLT3(ITD,F691L)
FLT3(K663Q) FLT3(N841I) FLT3(R834Q) FLT3-autoinhibited FLT4
FOXO3 FPR1 FPR3 FPRL1 FRK
FSHR FXR FYN G9a GABBR1-GABBR2
GAK GALR1 GALR2 GCGR GCN2(Kin.Dom.2,S808G)
GCN5L2 GHRHR GHR-JAK1 GHR-JAK2 GHSR
GHSR1b GIPR GLP GLP1R GLP2R
GNRHR GPBAR1 GPR1 GPR101 GPR103
GPR107 GPR109A GPR109B GPR119 GPR12
GPR120 GPR120S GPR123 GPR132 GPR135
GPR137 GPR139 GPR141 GPR142 GPR143
GPR146 GPR148 GPR149 GPR15 GPR150
GPR151 GPR152 GPR157 GPR161 GPR162
GPR17 GPR171 GPR173 GPR176 GPR18
GPR182 GPR20 GPR22 GPR23 GPR25
GPR26 GPR27 GPR3 GPR30 GPR31
GPR32 GPR35 GPR37 GPR37L1 GPR39
GPR4 GPR45 GPR50 GPR52 GPR55
GPR6 GPR61 GPR65 GPR75 GPR78
GPR79 GPR81 GPR83 GPR84 GPR85
GPR88 GPR92 GPR97 GR GRK1
GRK2 GRK3 GRK4 GRK7 GRM1
GRM2 GRM3 GRM4 GRM5 GRM6
GRPR GSK3A GSK3B HASPIN HCK
HCRTR1 HCRTR2 HIPK1 HIPK2 HIPK3
HIPK4 HitHunter® cAMP Assay for Biologics HitHunter® cAMP Assay for Small Molecules HPK1 HRH1
HRH2 HRH3 HRH4 HTR1A HTR1B
HTR1E HTR1F HTR2A HTR2B HTR2C
HTR2C(VGV) HTR2C(VNV) HTR2C(VSV) HTR5A HTR6
HTR7A HTR7B HTR7D HUNK ICK
IFNAR1/IFNAR2 IFNGR1/IFNGR2 IFNRL1/IL10RB IGF1R IKK-alpha
IKK-beta IKK-epsilon IL10RA/IL10RB IL11RA/IL6ST IL12RB1/IL12RB2
IL17RA/IL17RC IL17RD/TNFR2 IL18R1/IL18RAP IL1R1/IL1RAP IL1RL1/IL1RAP
IL20RA/IL10RB IL20RA/IL20RB IL21R/IL2RG IL22RA1/IL10RB IL23R/IL12RB1
IL27RA/IL6ST IL2RB/IL2RG IL2RB/IL2RG/IL2RA IL31RA/OSMRb IL3RA/CD131
IL4R/IL13RA1 IL4R/IL2RG IL5RA/CD131 IL6R/IL6ST IL7R/CRLF2
IL7R/IL2RG IL9R/IL2RG INSR INSRa INSRb
INSRR IRAK1 IRAK2 IRAK3 IRAK4
ITK IκB JAK1(JH1domain-catalytic) JAK1(JH2domain-pseudokinase) JAK2(JH1domain-catalytic)
JAK3 JAK3(JH1domain-catalytic) JNK1 JNK2 JNK3
KCNH2(G601S) KDR KDR/KDR Keap1-NRF2 KISS1R
KIT KIT(A829P) KIT(D816H) KIT(D816V) KIT(L576P)
KIT(V559D) KIT(V559D,T670I) KIT(V559D,V654A) KIT-autoinhibited LATS1
LATS2 LCK LGR4 LGR5 LGR6
LHCGR LIMK1 LIMK2 LKB1 LOK
LRRK2 LRRK2(G2019S) LTB4R LTK LXRα
LXRβ LXRβ-NCoR1 LYN LZK mADCYAP1R1
mADORA2B mADORA3 mADRA1B mAGTRL1 MAK
MAP3K1 MAP3K15 MAP3K2 MAP3K3 MAP3K4
MAP4K2 MAP4K3 MAP4K4 MAP4K5 MAPKAPK2
MAPKAPK5 MARK1 MARK2 MARK3 MARK4
MAST1 mAVPR2 mBRS3 MC1R MC3R
MC4R MC4R(T162I) mC5AR1 MC5R mCCKAR
mCCR1 mCCR2 mCCR3 mCCR4 mCCR5
mCCR6 mCCR7 mCCR8 mCCR9 MCHR1
MCHR2 MCL1-BIM mCMKLR1 mCNR1 mCNR2
mCRHR1 mCRTH2 mCX3CR1 mCXCR2 mCXCR3
mCXCR4 mCXCR5 mCXCR6 mCXCR7 mDRD5
mEBI2 mEDG1 mEDG3 mEDG5 mEDNRA
mEDNRB MEK1 MEK2 MEK3 MEK4
MEK5 MEK6 MELK MERTK MET
MET(M1250T) MET(Y1235D) mF2RL1 mFFAR1 mFPR1
mFPR2 mGALR1 mGALR2 mGCGR mGHSR
mGIPR mGLP1R mGLP1R-ADCY2 mGPR1 mGPR120
mGPR84 mHCRTR1 mHTR2A mHTR2C MINK
mINSRa mINSRb MKK7 MKNK1 MKNK2
MLCK MLK1 MLK2 MLK3 MLKL
MLKL(full-length) MLNR mLTB4R mMC3R mMC4R
mMC5R mMCHR1 mNPY1R mNPY2R mOPRD1
mOPRK1 mOPRM1 mOXTR mP2RY12 mP2RY6
mPPYR1 mPTAFR mPTGER4 mPTGIR MR
MRCKA MRCKB MRGPRD MRGPRE MRGPRF
MRGPRX1 MRGPRX2 MRGPRX4 mRHO(P23H) mRXFP1
mRXFP3 mRXFP4 mSSTR2 mSSTR5 MST1
MST1R MST2 MST3 MST4 mTAAR1
mTACR1 MTH1 MTNR1A MTNR1B MTOR
MUSK mUTR2 mVIPR1 MYLK MYLK2
MYLK4 MYO3A MYO3B NDR1 NDR2
NEK1 NEK10 NEK11 NEK2 NEK3
NEK4 NEK5 NEK6 NEK7 NEK9
NIK NIM1 NLK NMBR NMU1R
NPBWR1 NPBWR2 NPFFR1 NPR1 NPSR1b
NPY1R NPY2R NTSR1 OPN5 OPRD1
OPRK1 OPRL1 OPRM1 OSMR/IL6ST OSR1
OX40 OXER1 OXGR1 OXTR P2RY1
P2RY11 P2RY12 P2RY2 P2RY4 P2RY6
P2RY8 p38-alpha p38-beta p38-delta p38-gamma
P53 PAK1 PAK2 PAK3 PAK4
PAK6 PAK7 PASK PBRM1(2) PBRM1(5)
PCAF PCTK1 PCTK2 PCTK3 PD-1
PDGFRa PDGFRb PD-L1 PD-L1/PD-L1 PD-L2
PDPK1 PFCDPK1(P.falciparum) PFPK5(P.falciparum) PFTAIRE2 PFTK1
PHKG1 PHKG2 PI3Kδ PIK3C2B PIK3C2G
PIK3CA PIK3CA(C420R) PIK3CA(E542K) PIK3CA(E545A) PIK3CA(E545K)
PIK3CA(H1047L) PIK3CA(H1047Y) PIK3CA(I800L) PIK3CA(M1043I) PIK3CA(Q546K)
PIK3CB PIK3CD PIK3CG PIK4CB PIKFYVE
PIM1 PIM2 PIM3 PIP5K1A PIP5K1C
PIP5K2B PIP5K2C PKAC-alpha PKAC-alpha(L206R) PKAC-beta
PKMYT1 PKN1 PKN2 PKNB(M.tuberculosis) PLK1
PLK2 PLK3 PLK4 PPARα PPARγ
PPARδ PPYR1 PRKCD PRKCE PRKCH
PRKCI PRKCQ PRKD1 PRKD2 PRKD3
PRKG1 PRKG2 PRKR PRKX PRLHR
PRLR-JAK1 PRLR-JAK2 PRMT3 PROKR1 PROKR2
PRP4 PRα PRβ PTAFR PTGDR
PTGER1 PTGER2 PTGER3 PTGER4 PTGFR
PTGIR PTHR1 PTHR2 PYK2 QSK
RAF1 RANK-IκB RARα RARβ rCHRM4
rCNR2 rCRTH2 rDRD1 rDRD2L rDRD2S
rEDG5 RELA-IκB RET RET(A883F) RET(M918T)
RET(V804E) RET(V804L) RET(V804M) rFFAR1 rGPR120
rGPR35 rHTR2C rhTrkA-rhP75 RIOK1 RIOK2
RIOK3 RIPK1 RIPK1 RIPK2 RIPK3
RIPK3 RIPK4 RIPK5 ROCK1 ROCK2
rOPRM1 ROS1 rPROKR1 rPROKR2 RPS6KA4(Kin.Dom.1-N-terminal)
RPS6KA4(Kin.Dom.2-C-terminal) RPS6KA5(Kin.Dom.1-N-terminal) RPS6KA5(Kin.Dom.2-C-terminal) rPTGER4 RSK1(Kin.Dom.1-N-terminal)
RSK1(Kin.Dom.2-C-terminal) RSK2(Kin.Dom.1-N-terminal) RSK2(Kin.Dom.2-C-terminal) RSK3(Kin.Dom.1-N-terminal) RSK3(Kin.Dom.2-C-terminal)
RSK4(Kin.Dom.1-N-terminal) RSK4(Kin.Dom.2-C-terminal) rTAAR1 rTrkA-rP75 rVIPR1
RXFP1 RXFP2 RXFP3 RXFP4 RXRα
RXRγ S6K1 SBK1 SCTR sEDG5
SGK SgK110 SGK2 SGK3 SIK
SIK1 SIK2 SLK SMARCA2 SMARCA4
SMO(W535L) SNARK SNRK SRC SREBP2
SRMS SRPK1 SRPK2 SRPK3 SSTR1
SSTR2 SSTR3 SSTR4 SSTR5 STK16
STK33 STK35 STK36 STK39 SYK
TAAR1 TAAR5 TACR1 TACR2 TACR3
TAF1(2) TAF1L(2) TAK1 TAOK1 TAOK2
TAOK3 TBK1 TBXA2R TEC TESK1
TGFBR1 TGFBR1/ACVR2 TGFBR1/ACVR2B TGFBR1/TGFBR2 TGFBR1/TGFBR2/ENG
TGFBR2 THRα THRβ TIE1 TIE2
Tie2 TIM3/TIM3 TLK1 TLK2 TNIK
TNK1 TNK2 TNNI3K TORC1 TORC2
TPOR/TPOR TRHR TRIM24(Bromo.) TRIM24(PHD,Bromo.) TRIM33
TrkA TrkA-P75 TrkB TrkB-P75 TrkC
TrkC-P75 TRPM6 TSHR(L) TSSK1B TSSK3
TTK TXK TYK2 TYK2(JH1domain-catalytic) TYK2(JH2domain-pseudokinase)
TYRO3 ULK1 ULK2 ULK3 UTR2
VEGFR2 VIPR1 VIPR2 VISTA/VISTA VPS34
VRK2 WDR9(2) WEE1 WEE2 WNK1
WNK2 WNK3 WNK4 XBP1 XCR1
YANK1 YANK2 YANK3 YES YES1
YSK1 YSK4 ZAK ZAP70 β-Catenin