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Alphabetical Target List

AAK1 ABL1 ABL1(E255K)-phosphorylated ABL1(F317I)-nonphosphorylated ABL1(F317I)-phosphorylated
ABL1(F317L)-nonphosphorylated ABL1(F317L)-phosphorylated ABL1(H396P)-nonphosphorylated ABL1(H396P)-phosphorylated ABL1(M351T)-phosphorylated
ABL1(Q252H)-nonphosphorylated ABL1(Q252H)-phosphorylated ABL1(T315I)-nonphosphorylated ABL1(T315I)-phosphorylated ABL1(Y253F)-phosphorylated
ABL1-nonphosphorylated ABL1-phosphorylated ABL2 ACVR1 ACVR1B
ACVR1B/BMPR2 ACVR1C/ACVR2 ACVR1C/ACVR2B ACVR2/ACVR1 ACVR2A
ACVR2B ACVRL1 ACVRL1/ACVR2 ACVRL1/ACVR2B ACVRL1/BMPR2
ADCK3 ADCK4 ADCYAP1R1 ADORA1 ADORA2A
ADORA2B ADORA3 ADRA1A ADRA1B ADRA1D(82-572)
ADRA2A ADRA2B ADRA2C ADRB1 ADRB2
ADRB2(W158A) ADRB3 AGTR1 AGTRL1 AKT1
AKT2 AKT3 ALK ALK(1151Tins) ALK(C1156Y)
ALK(F1174L) ALK(L1196M) AMPK-alpha1 AMPK-alpha2 ANKK1
AR ARK5 ASK1 ASK2 ATAD2A
ATAD2B ATAD2B AURKA AURKB AURKC
AVPR1A AVPR1B AVPR2 AVPR2(S167T) AXL
BAI1 BAI2 BAI3 BAZ2A BAZ2A
BAZ2B BCL2-BAX BCL2-BIM BCL2L1-BAX BCL2L1-BIM
BDKRB1 BDKRB2 BIKE BLK BMPR1A
BMPR1A/ACVR2 BMPR1A/ACVR2B BMPR1A/BMPR2 BMPR1B BMPR1B/ACVR2
BMPR1B/ACVR2B BMPR1B/BMPR2 BMPR2 BMX BRAF
BRAF(V600E) BRD1 Brd2(1) BRD2(1,2) BRD2(2)
BRD3(1) BRD3(1) BRD3(1,2) BRD3(2) Brd4(1)
BRD4(1,2) BRD4(2) BRD4(full-length,short-iso.) Brd7 BRD8(1)
BRD8(2) BRD9 BrdT(1) BRDT(1,2) BRDT(2)
BRK BRPF1 BRPF3 BRPF3 BRS3
BRSK1 BRSK2 BRWD3(2) BTK BUB1
C3AR1 C5AR1 C5L2 CALCR CALCRL-RAMP1
CALCRL-RAMP2 CALCRL-RAMP3 CALCR-RAMP2 CALCR-RAMP3 CAMK1
CAMK1B CAMK1D CAMK1G CAMK2A CAMK2B
CAMK2D CAMK2G CAMK4 CAMKK1 CAMKK2
CASK CASR CCKAR CCKBR CCR1
CCR10 CCR2 CCR3 CCR4 CCR5
CCR6 CCR7 CCR8 CCR9 CCRL1
CCRL2 CD137 CD86 CDC25A CDC2L1
CDC2L2 CDC2L5 CDK1 CDK10 CDK11
CDK12 CDK2 CDK20 CDK3 CDK4
CDK4-cyclinD1 CDK4-cyclinD1(F93L) CDK4-cyclinD3 CDK5 CDK6
CDK7 CDK8 CDK9 CDKL1 CDKL2
CDKL3 CDKL5 CECR2 cEDG5 CFTR-ΔF508
cGPR91 CHEK1 CHEK2 CHRM1 CHRM2
CHRM3 CHRM4 CHRM5 cINSRa cINSRb
CIT c-KIT CLK1 CLK2 CLK3
CLK4 c-MET/c-MET CMKLR1 CNR1 CNR2
CREBBP c-Ret-GFRα1 c-Ret-GFRα2 CRHR1 CRHR2
CRTH2 CSF1R CSF1R/CSF1R CSF1R-autoinhibited CSF2RB/CSF2RA
CSF3R-JAK1 CSK CSNK1A1 CSNK1A1L CSNK1D
CSNK1E CSNK1G1 CSNK1G2 CSNK1G3 CSNK2A1
CSNK2A2 CTK CTLA4 CX3CR1 CXCR1
CXCR2 CXCR3 CXCR4 CXCR5 CXCR6
CXCR7 cyno CXCR1 cyno CXCR2 cyno GPR120 cyno MRGPRX2
CYSLTR2 DAPK1 DAPK2 DAPK3 DARC
DCAMKL1 DCAMKL2 DCAMKL3 DDR1 DDR2(T654M)
DLK DMPK DMPK2 DRAK1 DRAK2
DRD1 DRD2L DRD2S DRD3 DRD4
DRD5 DYRK1A DYRK1B DYRK2 EBI2
EDG1 EDG2 EDG3 EDG4 EDG5
EDG6 EDG7 EDNRA EDNRB EGFR
EGFR(E746-A750del) EGFR(G719C) EGFR(G719S) EGFR(L747-E749del, A750P) EGFR(L747-S752del, P753S)
EGFR(L747-T751del,Sins) EGFR(L858R) EGFR(L858R,T790M) EGFR(L861Q) EGFR(S752-I759del)
EGFR(T790M) EGFR/EGFR EGFR/ErbB2 EGFR/ErbB3 EIF2AK1
EP300 EP300 EPHA1 EPHA2 EPHA3
EphA4 EphA5 EPHA6 EphA7 EPHA8
EphB1 EphB2 EphB3 EphB4 EPHB6
EpoR/EpoR EpoR-JAK2 ErbB1 ERBB2 ErbB2/ErbB3
ErbB2/ErbB4 ErbB2-ErbB3 ERBB3 ErbB4 ErbB4/ErbB4
ERK1 ERK1(Q122L) ERK2 ERK3 ERK4
ERK5 ERK8 ERN1 ERRα ERα
F2R F2RL1 F2RL3 FAK FALZ
FALZ FER FES FFAR1 FFAR2
FFAR3 FGFR1 FGFR1-α-Klotho FGFR1-β-Klotho FGFR2
FGFR2(N550K) FGFR3 FGFR3(G380R)/FGFR3(G380R) FGFR3(G697C) FGFR3(K650E)
FGFR3(V555M) FGFR3/FGFR3 FGFR4 FGFR4 FGFR4-α-Klotho
FGFR4-β-Klotho FGR FLT1 FLT3 FLT3(D835H)
FLT3(D835V) FLT3(D835Y) FLT3(ITD) FLT3(ITD,D835V) FLT3(ITD,F691L)
FLT3(K663Q) FLT3(N841I) FLT3(R834Q) FLT3-autoinhibited FLT4
FOXO3 FPR1 FPR3 FPRL1 FRK
FSHR FXR FYN G9a GABBR1-GABBR2
GAK GALR1 GALR2 GCGR GCN2(Kin.Dom.2,S808G)
GCN5L2 GHRHR GHR-JAK1 GHR-JAK2 GHSR
GHSR1b GIPR GLP GLP1R GLP2R
GNRHR GPBAR1 GPR1 GPR101 GPR103
GPR107 GPR109A GPR109B GPR119 GPR12
GPR120 GPR120S GPR123 GPR132 GPR135
GPR137 GPR139 GPR141 GPR142 GPR143
GPR146 GPR148 GPR149 GPR15 GPR150
GPR151 GPR152 GPR157 GPR161 GPR162
GPR17 GPR171 GPR173 GPR176 GPR18
GPR182 GPR20 GPR22 GPR23 GPR25
GPR26 GPR27 GPR3 GPR30 GPR31
GPR32 GPR35 GPR37 GPR37L1 GPR39
GPR4 GPR45 GPR50 GPR52 GPR55
GPR6 GPR61 GPR65 GPR75 GPR78
GPR79 GPR81 GPR83 GPR84 GPR85
GPR88 GPR92 GPR97 GR GRK1
GRK2 GRK3 GRK4 GRK7 GRM1
GRM2 GRM3 GRM4 GRM5 GRM6
GRPR GSK3A GSK3B HASPIN HCK
HCRTR1 HCRTR2 HIPK1 HIPK2 HIPK3
HIPK4 HPK1 HRH1 HRH2 HRH3
HRH4 HTR1A HTR1B HTR1E HTR1F
HTR2A HTR2B HTR2C HTR2C(VGV) HTR2C(VNV)
HTR2C(VSV) HTR5A HTR6 HTR7A HTR7B
HTR7D HUNK ICK IFNAR1/IFNAR2 IFNGR1/IFNGR2
IFNRL1/IL10RB IGF1R IKK-alpha IKK-beta IKK-epsilon
IL10RA/IL10RB IL11RA/IL6ST IL12RB1/IL12RB2 IL17RA/IL17RC IL17RD/TNFR2
IL18R1/IL18RAP IL1R1/IL1RAP IL1RL1/IL1RAP IL20RA/IL10RB IL20RA/IL20RB
IL21R/IL2RG IL22RA1/IL10RB IL23R/IL12RB1 IL27RA/IL6ST IL2RB/IL2RG
IL2RB/IL2RG/IL2RA IL31RA/OSMRb IL3RA/CD131 IL4R/IL13RA1 IL4R/IL2RG
IL5RA/CD131 IL6R/IL6ST IL7R/CRLF2 IL7R/IL2RG IL9R/IL2RG
INSR INSRa INSRb INSRR IRAK1
IRAK2 IRAK3 IRAK4 ITK IκB
JAK1(JH1domain-catalytic) JAK1(JH2domain-pseudokinase) JAK2(JH1domain-catalytic) JAK3 JAK3(JH1domain-catalytic)
JNK1 JNK2 JNK3 KCNH2(G601S) KDR
KDR/KDR Keap1-NRF2 KISS1R KIT KIT(A829P)
KIT(D816H) KIT(D816V) KIT(L576P) KIT(V559D) KIT(V559D,T670I)
KIT(V559D,V654A) KIT-autoinhibited LATS1 LATS2 LCK
LGR4 LGR5 LGR6 LHCGR LIMK1
LIMK2 LKB1 LOK LRRK2 LRRK2(G2019S)
LTB4R LTK LXRα LXRβ LXRβ-NCoR1
LYN LZK mADCYAP1R1 mADORA2B mADORA3
mADRA1B mAGTRL1 MAK MAP3K1 MAP3K15
MAP3K2 MAP3K3 MAP3K4 MAP4K2 MAP4K3
MAP4K4 MAP4K5 MAPKAPK2 MAPKAPK5 MARK1
MARK2 MARK3 MARK4 MAST1 mAVPR2
mBRS3 MC1R MC3R MC4R MC4R(T162I)
mC5AR1 MC5R mCCKAR mCCR1 mCCR2
mCCR3 mCCR4 mCCR5 mCCR6 mCCR7
mCCR8 mCCR9 MCHR1 MCHR2 MCL1-BIM
mCMKLR1 mCNR1 mCNR2 mCRHR1 mCRTH2
mCX3CR1 mCXCR2 mCXCR3 mCXCR4 mCXCR5
mCXCR6 mCXCR7 mDRD5 mEBI2 mEDG1
mEDG3 mEDG5 mEDNRA mEDNRB MEK1
MEK2 MEK3 MEK4 MEK5 MEK6
MELK MERTK MET MET(M1250T) MET(Y1235D)
mF2RL1 mFFAR1 mFPR1 mFPR2 mGALR1
mGALR2 mGCGR mGHSR mGIPR mGLP1R
mGLP1R-ADCY2 mGPR1 mGPR120 mGPR84 mHCRTR1
mHTR2A mHTR2C MINK mINSRa mINSRb
MKK7 MKNK1 MKNK2 MLCK MLK1
MLK2 MLK3 MLKL MLKL(full-length) MLNR
mLTB4R mMC3R mMC4R mMC5R mMCHR1
mNPY1R mNPY2R mOPRD1 mOPRK1 mOPRM1
mOXTR mP2RY12 mP2RY6 mPPYR1 mPTAFR
mPTGER4 mPTGIR MR MRCKA MRCKB
MRGPRD MRGPRE MRGPRF MRGPRX1 MRGPRX2
MRGPRX4 mRHO(P23H) mRXFP1 mRXFP3 mRXFP4
mSSTR2 mSSTR5 MST1 MST1R MST2
MST3 MST4 mTAAR1 mTACR1 MTH1
MTNR1A MTNR1B MTOR MUSK mUTR2
mVIPR1 MYLK MYLK2 MYLK4 MYO3A
MYO3B NDR1 NDR2 NEK1 NEK10
NEK11 NEK2 NEK3 NEK4 NEK5
NEK6 NEK7 NEK9 NIK NIM1
NLK NMBR NMU1R NPBWR1 NPBWR2
NPFFR1 NPR1 NPSR1b NPY1R NPY2R
NTSR1 OPN5 OPRD1 OPRK1 OPRL1
OPRM1 OSMR/IL6ST OSR1 OX40 OXER1
OXGR1 OXTR P2RY1 P2RY11 P2RY12
P2RY2 P2RY4 P2RY6 P2RY8 p38-alpha
p38-beta p38-delta p38-gamma P53 PAK1
PAK2 PAK3 PAK4 PAK6 PAK7
PASK PBRM1(2) PBRM1(5) PCAF PCTK1
PCTK2 PCTK3 PD-1 PDGFRa PDGFRb
PD-L1 PD-L1/PD-L1 PD-L2 PDPK1 PFCDPK1(P.falciparum)
PFPK5(P.falciparum) PFTAIRE2 PFTK1 PHKG1 PHKG2
PI3Kδ PIK3C2B PIK3C2G PIK3CA PIK3CA(C420R)
PIK3CA(E542K) PIK3CA(E545A) PIK3CA(E545K) PIK3CA(H1047L) PIK3CA(H1047Y)
PIK3CA(I800L) PIK3CA(M1043I) PIK3CA(Q546K) PIK3CB PIK3CD
PIK3CG PIK4CB PIKFYVE PIM1 PIM2
PIM3 PIP5K1A PIP5K1C PIP5K2B PIP5K2C
PKAC-alpha PKAC-alpha(L206R) PKAC-beta PKMYT1 PKN1
PKN2 PKNB(M.tuberculosis) PLK1 PLK2 PLK3
PLK4 PPARα PPARγ PPARδ PPYR1
PRKCD PRKCE PRKCH PRKCI PRKCQ
PRKD1 PRKD2 PRKD3 PRKG1 PRKG2
PRKR PRKX PRLHR PRLR-JAK1 PRLR-JAK2
PRMT3 PROKR1 PROKR2 PRP4 PRα
PRβ PTAFR PTGDR PTGER1 PTGER2
PTGER3 PTGER4 PTGFR PTGIR PTHR1
PTHR2 PYK2 QSK RAF1 RANK-IκB
RARα RARβ rCHRM4 rCNR2 rCRTH2
rDRD1 rDRD2L rDRD2S rEDG5 RELA-IκB
RET RET(A883F) RET(M918T) RET(V804E) RET(V804L)
RET(V804M) rFFAR1 rGPR120 rGPR35 rHTR2C
rhTrkA-rhP75 RIOK1 RIOK2 RIOK3 RIPK1
RIPK1 RIPK2 RIPK3 RIPK3 RIPK4
RIPK5 ROCK1 ROCK2 rOPRM1 ROS1
rPROKR1 rPROKR2 RPS6KA4(Kin.Dom.1-N-terminal) RPS6KA4(Kin.Dom.2-C-terminal) RPS6KA5(Kin.Dom.1-N-terminal)
RPS6KA5(Kin.Dom.2-C-terminal) rPTGER4 RSK1(Kin.Dom.1-N-terminal) RSK1(Kin.Dom.2-C-terminal) RSK2(Kin.Dom.1-N-terminal)
RSK2(Kin.Dom.2-C-terminal) RSK3(Kin.Dom.1-N-terminal) RSK3(Kin.Dom.2-C-terminal) RSK4(Kin.Dom.1-N-terminal) RSK4(Kin.Dom.2-C-terminal)
rTAAR1 rTrkA-rP75 rVIPR1 RXFP1 RXFP2
RXFP3 RXFP4 RXRα RXRγ S6K1
SBK1 SCTR sEDG5 SGK SgK110
SGK2 SGK3 SIK SIK1 SIK2
SLK SMARCA2 SMARCA4 SMO(W535L) SNARK
SNRK SRC SREBP2 SRMS SRPK1
SRPK2 SRPK3 SSTR1 SSTR2 SSTR3
SSTR4 SSTR5 STK16 STK33 STK35
STK36 STK39 SYK TAAR1 TAAR5
TACR1 TACR2 TACR3 TAF1(2) TAF1L(2)
TAK1 TAOK1 TAOK2 TAOK3 TBK1
TBXA2R TEC TESK1 TGFBR1 TGFBR1/ACVR2
TGFBR1/ACVR2B TGFBR1/TGFBR2 TGFBR1/TGFBR2/ENG TGFBR2 THRα
THRβ TIE1 TIE2 Tie2 TIM3/TIM3
TLK1 TLK2 TNIK TNK1 TNK2
TNNI3K TORC1 TORC2 TPOR/TPOR TRHR
TRIM24(Bromo.) TRIM24(PHD,Bromo.) TRIM33 TrkA TrkA-P75
TrkB TrkB-P75 TrkC TrkC-P75 TRPM6
TSHR(L) TSSK1B TSSK3 TTK TXK
TYK2 TYK2(JH1domain-catalytic) TYK2(JH2domain-pseudokinase) TYRO3 ULK1
ULK2 ULK3 UTR2 VEGFR2 VIPR1
VIPR2 VISTA/VISTA VPS34 VRK2 WDR9(2)
WEE1 WEE2 WNK1 WNK2 WNK3
WNK4 XBP1 XCR1 YANK1 YANK2
YANK3 YES YES1 YSK1 YSK4
ZAK ZAP70 β-Catenin