| Biological Information | |
|---|---|
| Background Information: | K 252a is a fungal alkaloid and analog of staurosporine that is a potent, cell-permeable inhibitor of PKC (IC50=32.9nM), calcium/calmodulin-stimulated phosphodiesterases (IC50=1.3-2.9uM), MLCK (Ki=20nM), and receptor tyrosine kinases. Promotes myogenic differentiation, neuronal culture survival, and apoptosis, among other biological effects. Provided as 200μg of dry powder. |
| Target Name: | K 252a |
| Usage | |
| Product Type: | Control Ligands & Inhibitors |
| Application: | Drug Discovery & Development |
| Storage Conditions: | Store at -20°C. Please avoid multiple freeze/thaw cycles. |
| Usage Disclaimer: | These products may be covered by issued US and/or foreign patents, patent application and subject to Limited Use Label License. Please visit discoverx.com/license for a list of products that are governed by limited use label license terms and relevant patent and trademark information. |
| Additional Information | |
| Brand: | DiscoverX |
K 252a
K 252a is an inhibitor of PKC, MLCK, and other receptor tyrosine kinases. This product is provided as 200μg of dry powder.
Datasheets
92-1245 Datasheet
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