| Biological Information | |
|---|---|
| Background Information: | SR 49059 is an orally active synthetic small molecule that is a potent and selective inhibitor of the arginine vasopressin (AVP) V1a-receptor (Ki=1.1-6.3nM). AVP is an important hormone for circulatory and water homeostasis, as well as renal hemodynamic alterations, water retention, and cardiac remodeling in congestive heart failure. SR 49059 shows promise in platelet aggregation inhibition and treatment of Raynaud's disease, dysmenorrhea, and tocolysis. Provided as 1 mg of dry powder. |
| Target Name: | SR 49059 |
| Usage | |
| Product Type: | Control Ligands & Inhibitors |
| Application: | Drug Discovery & Development |
| Storage Conditions: | Store at 2-8°C. Please avoid multiple freeze/thaw cycles. |
| Usage Disclaimer: | These products may be covered by issued US and/or foreign patents, patent application and subject to Limited Use Label License. Please visit discoverx.com/license for a list of products that are governed by limited use label license terms and relevant patent and trademark information. |
| Additional Information | |
| Brand: | DiscoverX |
SR 49059
SR 49059 is an antagonist for AVPR1a, AVPR1b, and AVPR2. This product is provided as 1 mg of dry powder.
Datasheets
92-1279 Datasheet
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