A-674563 |
|
|
|
Yes |
|
AB-1010/Masitinib |
|
|
|
Yes |
|
ABT-869/Linifanib |
|
Yes |
Yes |
Yes |
FLT3, CSF1R, VEGFR2 |
AC220/Quizartinib |
Yes |
|
|
Yes |
FLT3 |
AG-013736/Axitinib |
|
|
|
Yes |
|
AMG-706/Motesanib |
|
Yes |
|
Yes |
VEGFR2, FLT1, FLT4, KIT |
AST-487 |
|
Yes |
|
Yes |
FLT3, KIT |
AT-7519 |
|
Yes |
|
Yes |
|
AZD-1152HQPA/Barasertib |
|
Yes |
|
Yes |
AURKB |
AZD-2171/Cediranib |
|
|
|
Yes |
|
AZD-6244/ARRY-886/Selumetinib |
|
|
|
Yes |
|
BI-2536 |
|
|
|
Yes |
|
BIBF-1120(derivative)/Nintedanib |
|
|
|
Yes |
|
BIBW-2992/Afatinib |
|
|
|
Yes |
|
BIRB-796/Doramapimod |
|
Yes |
Yes |
Yes |
p38-alpha |
BMS-345541 |
|
|
|
Yes |
|
BMS-387032/SNS-032 |
|
Yes |
|
Yes |
CDK2 |
BMS-540215/Brivanib |
|
|
|
Yes |
|
CEP-701/Lestaurtinib |
Yes |
|
|
Yes |
JAK2 |
CGP-52421 |
Yes |
|
|
|
FLT3 |
CHIR-258/TKI-258/Dovitinib |
|
Yes |
|
Yes |
FLT3, FGFR3 |
CHIR-265/RAF-265 |
|
Yes |
|
Yes |
BRAF, VEGFR2 |
CI-1033/Canertinib |
|
Yes |
Yes |
Yes |
EGFR, ERBB2 |
CI-1040 |
|
|
|
Yes |
|
CP-690550/tofacitinib |
|
Yes |
|
Yes |
JAK3 |
CP-724714 |
|
Yes |
|
|
ERBB2 |
Crizotinib |
|
|
|
Yes |
|
Dasatinib |
|
Yes |
|
Yes |
ABL1, SRC |
EKB-569 |
|
Yes |
Yes |
|
EGFR |
Erlotinib |
|
Yes |
Yes |
Yes |
EGFR |
EXEL-2880/GSK1363089/Foretinib |
|
|
|
Yes |
|
Flavopiridol/Alvocidib |
|
Yes |
Yes |
Yes |
CDK1,2,4, & CDK9 |
GDC-0879 |
|
|
|
Yes |
BRAF |
GDC-0941/Pictilisib |
|
|
|
Yes |
pan-PI3K |
Gefitinib |
|
Yes |
Yes |
Yes |
EGFR |
GSK-1838705A |
|
|
|
Yes |
|
GSK-461364A |
|
|
|
Yes |
|
GSK-690693 |
|
|
|
Yes |
|
GW-2580 |
|
Yes |
|
Yes |
CSF1R |
HKI-272/Neratinib |
|
|
|
Yes |
EGFR |
Imatinib |
|
Yes |
Yes |
Yes |
ABL1, KIT, PDGFRB |
INCB018424/Ruxolitinib |
|
|
|
Yes |
JAK1, JAK2 |
JNJ-28312141 |
|
|
|
Yes |
|
JNJ-7706621 |
|
Yes |
|
|
CDK2, CDK1, AURKB |
Ki-20227 |
|
|
|
Yes |
|
KW-2449 |
|
|
|
Yes |
|
Lapatinib/GW-2016 |
|
Yes |
Yes |
Yes |
EGFR, ERBB2 |
LY-317615/Enzastaurin |
|
|
|
Yes |
|
LY-333531/Ruboxistaurin |
|
Yes |
Yes |
Yes |
PRKCB1 |
MLN-120B |
|
|
|
Yes |
|
MLN-518/Tandutinib |
Yes |
Yes |
Yes |
Yes |
FLT3, KIT |
MLN-8054 |
|
Yes |
|
Yes |
AURKA |
Nilotinib/AMN107 |
|
|
|
Yes |
|
Pazopanib/GW-786034 |
|
Yes |
|
Yes |
FLT1, FLT4, PDGFRA, PDGFRB, VEGFR1, VEGFR2, VEGFR3 |
PD-173955 |
|
|
|
Yes |
|
PHA-665752 |
|
|
|
Yes |
|
PI-103 |
|
Yes |
|
Yes |
PIK3CA |
Midostaurin/PKC-412 |
Yes |
Yes |
Yes |
Yes |
FLT3, KIT |
PP-242 |
|
|
|
Yes |
|
PLX-4720 |
|
|
|
Yes |
|
R406/Tamatinib |
|
|
|
Yes |
|
R547 |
|
|
|
Yes |
|
Roscovitine/CYC202 |
|
Yes |
Yes |
|
CDK1, CDK2, CDK5 |
SB-202190 |
|
Yes |
Yes |
|
p38-alpha |
SB-203580 |
|
Yes |
Yes |
Yes |
p38-alpha |
SB-431542 |
|
Yes |
|
|
TGFBR1/ALK5, ACVR1B/ALK4 |
SGX-523 |
|
|
|
Yes |
|
SKI-606/Bosutinib |
|
|
|
Yes |
|
Sorafenib/BAY-43-9006 |
Yes |
Yes |
Yes |
Yes |
VEGFR2, BRAF |
SP600125 |
|
|
Yes |
|
JNK |
Staurosporine |
|
Yes |
Yes |
Yes |
PRKCH, Pan-inhibitor |
SU-14813 |
|
Yes |
|
Yes |
FLT1, FLT3, KIT, PDGFRB, VEGFR2 |
Sunitinib/SU-11248 |
Yes |
Yes |
Yes |
Yes |
KIT, FLT3, VEGFR2 |
TAE-684 |
|
|
|
Yes |
|
TG-101348/Fedratinib |
|
|
|
Yes |
|
TG-100-115 |
|
|
|
Yes |
|
Vatalanib/PTK-787 |
|
Yes |
Yes |
Yes |
VEGFR2 |
VX-680/MK-0457/Tozasertib |
|
Yes |
|
Yes |
AURKA, AURKB, AURKC |
VX-745 |
|
Yes |
Yes |
Yes |
p38-alpha |
ZD-6474/Vandetanib |
|
Yes |
Yes |
Yes |
VEGFR2, EGFR, RET |